Slow-binding inhibition of cholinesterases, pharmacological and toxicological relevance - ScienceDirect
Peptide Deformylase Inhibitors as Antibacterial Agents: Identification of VRC3375, a Proline-3-Alkylsuccinyl Hydroxamate Derivative, by Using an Integrated Combinatorial and Medicinal Chemistry Approach
Peptide Deformylase as an Antibacterial Drug Target: Target Validation and Resistance Development
Carmela GIGLIONE, Laboratory Head, PhD, Université Paris-Saclay, Paris
Inhibition and enzymatic reactions progress through an induced fit
Full article: Atomic level and structural understanding of natural ligands inhibiting Helicobacter pylori peptide deformylase through ligand and receptor based screening, SIFT, molecular dynamics and DFT – a structural computational approach
Full article: Atomic level and structural understanding of natural ligands inhibiting Helicobacter pylori peptide deformylase through ligand and receptor based screening, SIFT, molecular dynamics and DFT – a structural computational approach
PDF) Trapping Conformational States Along Ligand-Binding Dynamics of Peptide Deformylase: The Impact of Induced Fit on Enzyme Catalysis
Frédéric Dardel's research works Paris Descartes University, Paris and other places
PDF) Trapping Conformational States Along Ligand-Binding Dynamics of Peptide Deformylase: The Impact of Induced Fit on Enzyme Catalysis
A [(32)P]NAD(+)-based method to identify and quantitate long residence time enoyl-acyl carrier protein reductase inhibitors. - Abstract - Europe PMC